Labetalol hydrochloride
CAS Number: 32780-64-6
Molecular Mass: 364.9 g/mol
Formula: C19H25ClN2O3
Smiles: CC(CCc1ccccc1)NCC(O)c1ccc(O)c(C(N)=O)c1.Cl
Synonymes:
Labetalol hydrochloride, 32780-64-6, Labetalol HCL, Labrocol, ScH 15719W, AH 5158A, Ibidomide hydrochloride, Sch-15719W, 1GEV3BAW9J, AH-5158A, NSC-290312, DTXSID0044654, AH-5158A HYDROCHLORIDE, SCH-15719W HYDROCHLORIDE, DTXCID8024654, NSC290312, 5-(1-Hydroxy-2-((1-methyl-3-phenylpropyl)amino)ethyl)salicylamide monohydrochloride, Benzamide, 2-hydroxy-5-(1-hydroxy-2-((1-methyl-3-phenylpropyl)amino)ethyl)-, monohydrochloride, 5-[1-Hydroxy-2-[(1-methyl-3-phenylpropyl)amino]ethyl]salicylamide monohydrochloride, Labetalol Hydrocloride, Hydrochloride, Labetalol, RefChem:58511, Labetalol HCl in Dextrose, Labetalol HCl in Sodium Chloride, LABETALOL HYDROCHLORIDE IN DEXTROSE, LABETALOL HYDROCHLORIDE IN SODIUM CHLORIDE, 2-Hydroxy-5-((1RS)-1-hydroxy-2-((1RS)-1-methyl-3-phenylpropylamino)ethyl)benzamide monohydrochloride 2-Hydroxy-5-((1RS)-1-hydroxy-2-((1SR)-1-methyl-3-phenylpropylamino)ethyl)benzamide monohydrochloride, 251-211-1, Amipress, Normodyne, Presdate, Trandate, Labetalol (hydrochloride), 2-Hydroxy-5-(1-hydroxy-2-((4-phenylbutan-2-yl)amino)ethyl)benzamide hydrochloride, Benzamide,2-hydroxy-5-[1-hydroxy-2-[(1-methyl-3-phenylpropyl)amino]ethyl]-, hydrochloride(1:1), MFCD00057663, 72487-34-4, MLS000069666, 2-hydroxy-5-[1-hydroxy-2-(4-phenylbutan-2-ylamino)ethyl]benzamide, hydrochloride, Labetalol (hydrochloride) (Standard), AH-5158 hydrochloride, Sch-15719W, Pressalolo, SMR000058463, Ipolab, rac-Labetalol Hydrochloride, 2-hydroxy-5-[1-hydroxy-2-(4-phenylbutan-2-ylamino)ethyl]benzamide hydrochloride, 5-(1-Hydroxy-2-((1-methyl-3-phenylpropyl)amino)ethyl)salicylamide hydrochloride, 5-[1-Hydroxy-2-[(1-methyl-3-phenylpropyl)amino]ethyl]salicylamide hydrochloride, 2-Hydroxy-5-[1-hydroxy-2-[(1-methyl-3-phenylpropyl)amino]ethyl]benzamide hydrochloride, CCRIS 1086, SR-01000000209, EINECS 251-211-1, UNII-1GEV3BAW9J, NSC 290312, 32780-64-6 (HCl), 2-hydroxy-5-(1-hydroxy-2-(4-phenylbutan-2-ylamino)ethyl)benzamide hydrochloride, 2-Hydroxy-5-(1-hydroxy-2-[(1-methyl-3-phenylpropyl)amino]ethyl)benzamide hydrochloride, Normodyne (TN), Trandate (TN), Prestwick_290, EINECS 276-694-6, Labeolol hydrochloride, Labetalol hydrochloride [USAN:USP:JAN], La.beta.lol hydrochloride, Opera_ID_1625, Benzamide,monohydrochloride, NCGC00016810-01, Salicylamide, hydrochloride, Labetalol hydrochloride CRS, CAS-32780-64-6, Salicylamide, 5-(1-hydroxy-2-((1-methyl-3-phenylpropyl)amino)ethyl)-, hydrochloride, SCHEMBL41230, MLS001148626, MLS002222197, SPECTRUM1503243, CHEBI:6344, orb1310699, CHEMBL1200323, SCHEMBL29710409, HY-B1108R, GLXC-06704, HMS1568H16, HMS1922M13, HMS5083I05, MSK000466A, Pharmakon1600-01503243, EX-A4940, HY-B1108, LABETALOL HYDROCHLORIDE [MI], Tox21_110623, Tox21_302725, Tox21_500687, CCG-40314, EBC-80148, Labetalol hydrochloride (JP18/USP), LABETALOL HYDROCHLORIDE [JAN], NSC758438, s4291, LABETALOL HYDROCHLORIDE [USAN], AKOS015895575, AC-1389, AH-5158, CS-4706, FL61512, LABETALOL HYDROCHLORIDE [MART.], LABETALOL HYDROCHLORIDE [VANDF], LP00687, MSK000466A-1000M, NC00571, NSC-758438, SS-4219, LABETALOL HYDROCHLORIDE [USP-RS], LABETALOL HYDROCHLORIDE [WHO-DD], NCGC00094044-01, NCGC00094044-02, NCGC00094044-03, NCGC00094044-04, NCGC00094044-05, NCGC00256847-01, NCGC00261372-01, (R*,R*)-(1)-5-(1-Hydroxy-2-((1-methyl-3-phenylpropyl)amino)ethyl)salicylamide monohydrochloride, DB-048265, CS-0694914, EU-0100687, LABETALOL HYDROCHLORIDE [ORANGE BOOK], NS00087824, SW196595-3, LABETALOL HYDROCHLORIDE [EP MONOGRAPH], D00600, LABETALOL HYDROCHLORIDE [USP MONOGRAPH], Labetalol hydrochloride, >98% (TLC), powder, NORMOZIDE COMPONENT LABETALOL HYDROCHLORIDE, SR-01000000209-2, SR-01000000209-7, Q27252396, Labetalol hydrochloride Solution in Methanol, 1000ug/mL, 2-Hydroxy-5-(1-hydroxy-2-((4-phenylbutan-2-yl)amino)ethyl)benzamide HCl, Labetalol hydrochloride, European Pharmacopoeia (EP) Reference Standard, Labetalol hydrochloride, United States Pharmacopeia (USP) Reference Standard, 2-hydroxy-5-[1-hydroxy-2-[(1-methyl-3-phenyl-propyl)amino]ethyl]benzamide, hydrochloride, Labetalol Hydrochloride, Pharmaceutical Secondary Standard, Certified Reference Material, (r*,r*)-( inverted exclamation markA)-5-[1-Hydroxy-2-[(1-methyl-3-phenylpropyl)amino]ethyl]salicylamide monohydrochloride, (R,R)-Dilevalol.HCl, 2-hydroxy-5-[(1R)-1-hydroxy-2-{[(1R)-1-methyl-3-phenylpropyl]amino}ethyl]benzamide hydrochloride, Dilevalol hydrochloride, (R,R)-Dilevalol hydrochloride, (-)-2-hydroxy-5-<(R)-1-hydroxy-2-<(R)-(1-methyl-3-phenylpropyl)amino>et, 2-Hydroxy-5-{1-hydroxy-2-[(4-phenylbutan-2-yl)amino]ethyl}benzamide--hydrogen chloride (1/1), Benzamide, 2-hydroxy-5-[1-hydroxy-2-[(1-methyl-3-phenylpropyl)amino]ethyl]-, hydrochloride (1:1), Mixture of 4 stereoisomers of 2-hydroxy-5-[1-hydroxy2-[(1-methyl-3-phenylpropyl)amino]ethyl]benzamide hydrochloride
Bioactivity: -
Solubility in Different Solvents
| Solvent | Temperature [K] | Crystal form | Solubility [mg/mL] | Reference |
|---|---|---|---|---|
| 1-Butanol | 288.15 | - | 1.542 | [334] |
| 1-Butanol | 293.15 | - | 1.862 | [334] |
| 1-Butanol | 298.15 | - | 2.243 | [334] |
| 1-Butanol | 303.15 | - | 2.667 | [334] |
| 1-Butanol | 308.15 | - | 3.178 | [334] |
| 1-Butanol | 313.15 | - | 3.785 | [334] |
| 1-Butanol | 318.15 | - | 4.52 | [334] |
| 1-Butanol | 323.15 | - | 5.275 | [334] |
| 1-Butanol | 328.15 | - | 6.293 | [334] |
| 1-Propanol | 288.15 | - | 2.345 | [334] |
| 1-Propanol | 293.15 | - | 2.83 | [334] |
| 1-Propanol | 298.15 | - | 3.45 | [334] |
| 1-Propanol | 303.15 | - | 4.067 | [334] |
| 1-Propanol | 308.15 | - | 4.8 | [334] |
| 1-Propanol | 313.15 | - | 5.792 | [334] |
| 1-Propanol | 318.15 | - | 6.859 | [334] |
| 1-Propanol | 323.15 | - | 8.198 | [334] |
| 1-Propanol | 328.15 | - | 9.148 | [334] |
| 2-Butanol | 288.15 | - | 0.6664 | [334] |
| 2-Butanol | 293.15 | - | 0.8378 | [334] |
| 2-Butanol | 298.15 | - | 1.098 | [334] |
| 2-Butanol | 303.15 | - | 1.32 | [334] |
| 2-Butanol | 308.15 | - | 1.607 | [334] |
| 2-Butanol | 313.15 | - | 2.002 | [334] |
| 2-Butanol | 318.15 | - | 2.486 | [334] |
| 2-Butanol | 323.15 | - | 3.091 | [334] |
| 2-Butanol | 328.15 | - | 3.757 | [334] |
| Ethanol | 288.15 | - | 7.801 | [334] |
| Ethanol | 293.15 | - | 9.081 | [334] |
| Ethanol | 298.15 | - | 10.6 | [334] |
| Ethanol | 303.15 | - | 12.27 | [334] |
| Ethanol | 308.15 | - | 13.68 | [334] |
| Ethanol | 313.15 | - | 15.51 | [334] |
| Ethanol | 318.15 | - | 17.56 | [334] |
| Ethanol | 323.15 | - | 21.2 | [334] |
| Ethanol | 328.15 | - | 23.83 | [334] |
| Ethyl acetate | 288.15 | - | 0.4355 | [334] |
| Ethyl acetate | 293.15 | - | 0.608 | [334] |
| Ethyl acetate | 298.15 | - | 0.8781 | [334] |
| Ethyl acetate | 303.15 | - | 1.111 | [334] |
| Ethyl acetate | 308.15 | - | 1.484 | [334] |
| Ethyl acetate | 313.15 | - | 1.927 | [334] |
| Ethyl acetate | 318.15 | - | 2.483 | [334] |
| Ethyl acetate | 323.15 | - | 2.945 | [334] |
| Ethyl acetate | 328.15 | - | 3.872 | [334] |
| Isobutanol | 288.15 | - | 0.5396 | [334] |
| Isobutanol | 293.15 | - | 0.7266 | [334] |
| Isobutanol | 298.15 | - | 1.01 | [334] |
| Isobutanol | 303.15 | - | 1.275 | [334] |
| Isobutanol | 308.15 | - | 1.67 | [334] |
| Isobutanol | 313.15 | - | 2.17 | [334] |
| Isobutanol | 318.15 | - | 2.809 | [334] |
| Isobutanol | 323.15 | - | 3.762 | [334] |
| Isobutanol | 328.15 | - | 4.81 | [334] |
| Isopropanol | 288.15 | - | 0.528 | [334] |
| Isopropanol | 293.15 | - | 0.7824 | [334] |
| Isopropanol | 298.15 | - | 1.2 | [334] |
| Isopropanol | 303.15 | - | 1.675 | [334] |
| Isopropanol | 308.15 | - | 2.31 | [334] |
| Isopropanol | 313.15 | - | 3.15 | [334] |
| Isopropanol | 318.15 | - | 4.572 | [334] |
| Isopropanol | 323.15 | - | 6.46 | [334] |
| Isopropanol | 328.15 | - | 8.911 | [334] |
| Methanol | 288.15 | - | 80.73 | [334] |
| Methanol | 293.15 | - | 91.91 | [334] |
| Methanol | 298.15 | - | 103.3 | [334] |
| Methanol | 303.15 | - | 117.0 | [334] |
| Methanol | 308.15 | - | 129.3 | [334] |
| Methanol | 313.15 | - | 144.8 | [334] |
| Methanol | 318.15 | - | 162.0 | [334] |
| Methanol | 323.15 | - | 180.9 | [334] |
| Methanol | 328.15 | - | 201.3 | [334] |
| Water | 288.15 | - | 14.4 | [334] |
| Water | 293.15 | - | 18.17 | [334] |
| Water | 298.15 | - | 23.86 | [334] |
| Water | 303.15 | - | 29.28 | [334] |
| Water | 308.15 | - | 34.69 | [334] |
| Water | 313.15 | - | 42.7 | [334] |
| Water | 318.15 | - | 53.49 | [334] |
| Water | 323.15 | - | 67.67 | [334] |
| Water | 328.15 | - | 81.99 | [334] |
Molecule 3D descriptors
| Descriptor | Value |
|---|---|
| PMI1 | 675.2911 |
| PMI2 | 8058.3354 |
| PMI3 | 8471.8649 |
| NPR1 | 0.0797 |
| NPR2 | 0.9512 |
| RadiusOfGyration | 4.8557 |
| InertialShapeFactor | 0.0014 |
| Eccentricity | 0.9968 |
| Asphericity | 0.7801 |
| SpherocityIndex | 0.0716 |
| PBF | 0.5928 |